Benjamin F. Cravatt

ChemistryBiochemistry, Genetics and Molecular Biology

Pilot corpus only

This score is computed over theSindex pilot corpus and does not cover the full scientific literature. Scores are relative to papers we have ingested — papers, authors, and institutions outside the pilot are not represented. Methodology.

Top 100%percentile

0Author DataRank

Indexed papers

0in pilot corpus

datarank_citation_only_1hop_v6· scope data_onlyMethodology

Papers

Driven by 86 papers. Top paper: “Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries”.

Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries

Nature Biotechnology(2021)10.1038/s41587-020-00778-3

N/A

0.873DataRank · unranked

335 citations

Dylan C. Mitchell, Devin K. Schweppe, Ajami Gikandi, David P. Nusinow, Nathan J. Bulloch +7 more

In situ identification of cellular drug targets in mammalian tissue

Cell(2022)10.1016/j.cell.2022.03.040

N/A

0.650DataRank · unranked

75 citations

Michael A. Schafroth, Daisuke Ogasawara, Yu Wang, Victoria Nudell, Neeraj K. Lal +9 more

Single-Cell Profiling and SCOPE-Seq Reveal Lineage Dynamics of Adult Ventricular-Subventricular Zone Neurogenesis and NOTUM as a Key Regulator

Cell Reports(2020)10.1016/j.celrep.2020.107805

N/A

0.635DataRank · unranked

68 citations

N. Sumru Bayın, Jinzhou Yuan, Zhouzerui Liu, Radu M. Suciu, Micah J. Niphakis +6 more

Chemical Proteomic Discovery of Isotype‐Selective Covalent Inhibitors of the RNA Methyltransferase NSUN2

Angewandte Chemie International Edition(2023)10.1002/anie.202311924

N/A

0.612DataRank · unranked

58 citations

Jan G. Felber, Zhongyu Zou, Evert Njomen, Jarrett R. Remsberg, Daisuke Ogasawara +7 more

Multi-tiered chemical proteomic maps of tryptoline acrylamide–protein interactions in cancer cells

Nature Chemistry(2024)10.1038/s41557-024-01601-1

N/A

0.606DataRank · unranked

56 citations

Rachel E. Hayward, Kristen E. DeMeester, Daisuke Ogasawara, Melissa M. Dix, Tracey Nguyen +6 more

Depletion of creatine phosphagen energetics with a covalent creatine kinase inhibitor

Nature Chemical Biology(2023)10.1038/s41589-023-01273-x

N/A

0.584DataRank · unranked

48 citations

Wenzhi Ji, Mengyang Fan, Shan Lin, Hyuk‐Soo Seo, Ekaterina V. Vinogradova +15 more

ABHD4-dependent developmental anoikis safeguards the embryonic brain

Nature Communications(2020)10.1038/s41467-020-18175-4

N/A

0.520DataRank · unranked

31 citations

Zsolt Lele, Miklós Zöldi, Vivien Miczán, Fruzsina Mógor, Gabriel M. Simon +5 more

Assigning functionality to cysteines by base editing of cancer dependency genes

bioRxiv (Cold Spring Harbor Laboratory)(2022)10.1101/2022.11.17.516964

N/A

0.487DataRank · unranked

9 citations

Jarrett R. Remsberg, Sang Joon Won, Kevin T. Zhao, Tony P. Huang, Bingwen Lu +4 more

Development of a highly-specific 18F-labeled irreversible positron emission tomography tracer for monoacylglycerol lipase mapping

Acta Pharmaceutica Sinica B(2021)10.1016/j.apsb.2021.01.021

N/A

0.425DataRank · unranked

16 citations

Wakana Mori, Jian Rong, Michael A. Schafroth, Tuo Shao, Richard Van +17 more

Cysteine allostery and autoinhibition govern human STING oligomer functionality

Nature Chemical Biology(2025)10.1038/s41589-025-01951-y

N/A

0.406DataRank · unranked

14 citations

Xujun Cao, Sabrina L. Ergun, Evert Njomen, Stephen R. Lynch, Christopher Ritchie +3 more

Covalent Targeting As a Common Mechanism for Inhibiting NLRP3 Inflammasome Assembly

ACS Chemical Biology(2024)10.1021/acschembio.3c00330

N/A

0.406DataRank · unranked

14 citations

Jie Sun, Kayla Nutsch, Jessica D. Rosarda, Thu Nguyen, Chloris Li-Ma +9 more

Chemical proteomic analysis of palmostatin beta-lactone analogs that affect N-Ras palmitoylation

Bioorganic & Medicinal Chemistry Letters(2021)10.1016/j.bmcl.2021.128414

N/A

0.406DataRank · unranked

8 citations

Irungu K. Luvaga, Akram Hazeen, Chulangani Weerasooriya, Stewart K. Richardson, Ari J. Firestone +4 more

Proteomic discovery of chemical probes that perturb protein complexes in human cells

bioRxiv (Cold Spring Harbor Laboratory)(2022)10.1101/2022.12.12.520090

N/A

0.373DataRank · unranked

11 citations

Jarrett R. Remsberg, Martin G. Jaeger, Katherine Rothamel, Hsuan-Lin Her, Kristen E. DeMeester +30 more

Chemical proteomic identification of functional cysteines with atypical electrophile reactivities

Tetrahedron Letters(2021)10.1016/j.tetlet.2021.152861

N/A

0.330DataRank · unranked

8 citations

Vincent M. Crowley, Radu M. Suciu, Dale L. Boger, Benjamin F. Cravatt, K. Litwin

Mapping cellular targets of covalent cancer drugs in the entire mammalian body

Cell(2025)10.1016/j.cell.2025.11.030

N/A

0.292DataRank · unranked

6 citations

Verina H. Leung, Cailynn C. Wang, Ahmadreza Attarpour, Anthony Rinaldi, Hanbing Shen +14 more

Simple, Enantiocontrolled Azetidine Library Synthesis via Strain Release Functionalization of 1-Azabicyclobutanes

ChemRxiv(2024)10.26434/chemrxiv-2024-cmvd4

N/A

0.208DataRank · unranked

3 citations

Molhm Nassir, Hayden A. Sharma, Nathanyal J. Truax, Nicholas Raheja, Ty M. Thompson +5 more

A cold-inducible phospholipid—protein interaction in brown fat mitochondria optimizes thermogenic capacity

bioRxiv (Cold Spring Harbor Laboratory)(2025)10.1101/2025.05.15.654206

N/A

0.104DataRank · unranked

1 citations

Marc J. Tol, Christian Rocha-Roa, Matthew J. Jellinek, Liujuan Cui, Aaron Bender +23 more

Prolyl endopeptidase-like is a (thio)esterase involved in mitochondrial respiratory chain function

iScience(2021)10.1016/j.isci.2021.103460

N/A

0DataRank · unranked

23 citations

Molly T. McDevitt, Joél Smet, Brendan J. Floyd, Maxime Verschoore, María J. Marcaida +17 more

Selective inhibition of monoacylglycerol lipase is associated with passive coping behavior and attenuation of stress-induced dopamine release in the medial prefrontal cortex

Neurobiology of Stress(2021)10.1016/j.ynstr.2021.100293

N/A

0DataRank · unranked

19 citations

Ilham Polis, David G. Stouffer, Benjamin F. Cravatt, Marisa Roberto, Rémi Martin‐Fardon +4 more

Multiplexed proteomic profiling of cysteine reactivity and ligandability in human T cells

STAR Protocols(2021)10.1016/j.xpro.2021.100458

N/A

0DataRank · unranked

14 citations

Benjamin F. Cravatt, Ekaterina V. Vinogradova

Refinement of covalent EGFR inhibitor AZD9291 to eliminate off-target activity

Tetrahedron Letters(2021)10.1016/j.tetlet.2021.153178

N/A

0DataRank · unranked

10 citations

Balyn W. Zaro, Melissa M. Dix, Benjamin F. Cravatt, Chi‐Huey Wong, Elise Bouffard

Publisher Correction: A proteome-wide atlas of lysine-reactive chemistry

Nature Chemistry(2021)10.1038/s41557-021-00823-x

N/A

0DataRank · unranked

3 citations

Madeline E. Kavanagh, Taka-Aki Ichu, Michael R. Lazear, Yongfeng Tao, Vincent M. Crowley +9 more

LPCAT3 Inhibitors Remodel the Polyunsaturated Phospholipid Content of Human Cells and Protect from Ferroptosis

ACS Chemical Biology(2022)10.1021/acschembio.2c00317

N/A

0DataRank · unranked

151 citations

Taka-Aki Ichu, Natalia Milosevich, Bruno Melillo, Michael A. Schafroth, Yuka Otsuka +4 more

Targeted Protein Degradation by Electrophilic PROTACs that Stereoselectively and Site-Specifically Engage DCAF1

Journal of the American Chemical Society(2022)10.1021/jacs.2c08964

N/A

0DataRank · unranked

133 citations

David Remillard, Ekaterina V. Vinogradova, Minoru Yokoyama, Sofia Banchenko, David Schwefel +5 more

Stereochemical diversity as a source of discovery in chemical biology

Current Research in Chemical Biology(2022)10.1016/j.crchbi.2022.100028

N/A

0DataRank · unranked

81 citations

Nathalie Ropek, Bruno Melillo, Stuart L. Schreiber, Benjamin F. Cravatt, Ekaterina V. Vinogradova +1 more

Selective inhibitors of SARM1 targeting an allosteric cysteine in the autoregulatory ARM domain

Proceedings of the National Academy of Sciences(2022)10.1073/pnas.2208457119

N/A

0DataRank · unranked

78 citations

Elisa Merlini, Carlos Guijas, Kristen E. DeMeester, Evert Njomen, Ellen M. Kozina +9 more

Hippo pathway regulation by phosphatidylinositol transfer protein and phosphoinositides

Nature Chemical Biology(2022)10.1038/s41589-022-01061-z

N/A

0DataRank · unranked

66 citations

Vivian Fu, Guangbo Liu, Tracy Tang, Andrei W. Konradi, Xiao Peng +9 more

Accelerated lysine metabolism conveys kidney protection in salt-sensitive hypertension

Nature Communications(2022)10.1038/s41467-022-31670-0

N/A

0DataRank · unranked

65 citations

Oleg Palygin, Ashraf El‐Meanawy, Xavier Domingo-Almenara, Amelia Palermo, Lashodya V. Dissanayake +20 more

Chemoproteomics‐Enabled Identification of 4‐Oxo‐β‐Lactams as Inhibitors of Dipeptidyl Peptidases 8 and 9

Angewandte Chemie International Edition(2022)10.1002/anie.202210498

N/A

0DataRank · unranked

13 citations

B. Ross, Lorenz Fehr, Oguz Bolgi, Svenja Wöhrle, Kenneth M. Lum +13 more

Chemoproteomik‐basierte Identifikation von 4‐Oxo‐β‐lactamen als Inhibitoren der Dipeptidylpeptidasen 8 und 9

Angewandte Chemie(2022)10.1002/ange.202210498

N/A

0DataRank · unranked

1 citations

B. Ross, Lorenz Fehr, Oguz Bolgi, Svenja Wöhrle, Kenneth M. Lum +13 more

TMEM164 is an acyltransferase that forms ferroptotic polyunsaturated ether phospholipids

bioRxiv (Cold Spring Harbor Laboratory)(2022)10.1101/2022.07.06.498872

N/A

0DataRank · unranked

4 citations

Timothy B. Ware, Haoxin Li, J. Fernando Bazán, Benjamin F. Cravatt, Alex Reed

Collateral lethality between HDAC1 and HDAC2 exploits cancer-specific NuRD complex vulnerabilities

bioRxiv (Cold Spring Harbor Laboratory)(2022)10.1101/2022.05.30.493851

N/A

0DataRank · unranked

2 citations

David Remillard, Ugoma Onubogu, Barbara Karakyriakou, Joshua N. Asiaban, Anissa R. Ramos +7 more

The metabolite α-ketobutyrate increases health and life spans by activating AMPK

bioRxiv (Cold Spring Harbor Laboratory)(2022)10.1101/2022.10.10.511641

N/A

0DataRank · unranked

0 citations

Brett Lomenick, Min Chai, Wilson Huang, Jessie Chu, Laurent Vergnes +23 more

Proteomic discovery of chemical probes that perturb protein complexes in human cells

Molecular Cell(2023)10.1016/j.molcel.2023.03.026

N/A

0DataRank · unranked

94 citations

Jarrett R. Remsberg, Martin G. Jaeger, Katherine Rothamel, Hsuan-Lin Her, Kristen E. DeMeester +30 more

Remodeling oncogenic transcriptomes by small molecules targeting NONO

Nature Chemical Biology(2023)10.1038/s41589-023-01270-0

N/A

0DataRank · unranked

87 citations

Seong Joo Koo, Garrett L. Lindsey, Hsuan-Lin Her, Steven M. Blue, Haoxin Li +7 more

Assigning functionality to cysteines by base editing of cancer dependency genes

Nature Chemical Biology(2023)10.1038/s41589-023-01428-w

N/A

0DataRank · unranked

63 citations

Tiantai Ma, Jarrett R. Remsberg, Sang Joon Won, Kristen E. DeMeester, Evert Njomen +11 more

TMEM164 is an acyltransferase that forms ferroptotic C20:4 ether phospholipids

Nature Chemical Biology(2023)10.1038/s41589-022-01253-7

N/A

0DataRank · unranked

58 citations

Timothy B. Ware, Haoxin Li, J. Fernando Bazán, Benjamin F. Cravatt, Alex Reed

Collateral lethality between HDAC1 and HDAC2 exploits cancer-specific NuRD complex vulnerabilities

Nature Structural & Molecular Biology(2023)10.1038/s41594-023-01041-4

N/A

0DataRank · unranked

34 citations

David Remillard, Ugoma Onubogu, Barbara Karakyriakou, Joshua N. Asiaban, Anissa R. Ramos +10 more

Activity‐Based Protein Profiling – Finding General Solutions to Specific Problems

Israel Journal of Chemistry(2023)10.1002/ijch.202300029

N/A

0DataRank · unranked

32 citations

Benjamin F. Cravatt

Sexually dimorphic effects of monoacylglycerol lipase inhibitor MJN110 on stress‐related behaviour and drinking in Marchigian Sardinian alcohol‐preferring rats

British Journal of Pharmacology(2023)10.1111/bph.16197

N/A

0DataRank · unranked

14 citations

Bryan Cruz, Hannah C. Feldman, R. W. Bullard, P Bianchi, Luis A. Natividad +5 more

Comprehensive Mapping of Electrophilic Small Molecule-Protein Interactions in Human Cells

ChemRxiv(2023)10.26434/chemrxiv-2023-s446n

N/A

0DataRank · unranked

13 citations

Evert Njomen, Rachel Hayward, Kristen E. DeMeester, Daisuke Ogasawara, Melissa M. Dix +6 more

Attenuating ABHD17 isoforms augments the S -acylation and function of NOD2 and a subset of Crohn’s disease-associated NOD2 variants

bioRxiv (Cold Spring Harbor Laboratory)(2023)10.1101/2023.12.20.572362

N/A

0DataRank · unranked

6 citations

Noah R. Martin, Micah J. Niphakis, Benjamin F. Cravatt, Gregory D. Fairn, Charneal L. Dixon

Three-dimensional bioprinted glioblastoma microenvironments model cellular dependencies and immune interactions

Cell Research(2020)10.1038/s41422-020-0338-1

N/A

0DataRank · unranked

282 citations

Qi Xie, Ryan C. Gimple, Zheng Zhong, Trevor Tam, Jing Tian +24 more

Glutathione supports lipid abundance in vivo

bioRxiv (Cold Spring Harbor Laboratory)(2023)10.1101/2023.02.10.524960

N/A

0DataRank · unranked

3 citations

Emily Tuttle, Nathan P. Ward, Yun Pyo Kang, Yumi Kim, Madeline E. Kavanagh +33 more

Chemical Proteomic Discovery of Isotype‐Selective Covalent Inhibitors of the RNA Methyltransferase NSUN2

Angewandte Chemie(2023)10.1002/ange.202311924

N/A

0DataRank · unranked

0 citations

Jan G. Felber, Zhongyu Zou, Evert Njomen, Jarrett R. Remsberg, Daisuke Ogasawara +7 more

Ligand discovery by activity-based protein profiling

Cell chemical biology(2024)10.1016/j.chembiol.2024.08.006

N/A

0DataRank · unranked

69 citations

Benjamin F. Cravatt, Micah J. Niphakis

Glutathione synthesis in the mouse liver supports lipid abundance through NRF2 repression

Nature Communications(2024)10.1038/s41467-024-50454-2

N/A

0DataRank · unranked

54 citations

Emily Tuttle, Nathan P. Ward, Yun Pyo Kang, Yumi Kim, Madeline E. Kavanagh +33 more

Proteomic Ligandability Maps of Spirocycle Acrylamide Stereoprobes Identify Covalent ERCC3 Degraders

Journal of the American Chemical Society(2024)10.1021/jacs.3c13448

N/A

0DataRank · unranked

40 citations

Jarrett R. Remsberg, Haoxin Li, Evert Njomen, Kristen E. DeMeester, Yongfeng Tao +9 more

Redirecting the pioneering function of FOXA1 with covalent small molecules

Molecular Cell(2024)10.1016/j.molcel.2024.09.024

N/A

0DataRank · unranked

36 citations

Yuxiang Zhang, Christopher J. Reinhardt, Lauren M Hargis, Nicole S. MacRae, Kristen E. DeMeester +6 more

Chemical tools to expand the ligandable proteome: Diversity-oriented synthesis-based photoreactive stereoprobes

Cell chemical biology(2024)10.1016/j.chembiol.2024.10.005

N/A

0DataRank · unranked

26 citations

David B. Konrad, Zher Yin Tan, Kimberly L. Carey, Jessica Y. Luo, Sang Joon Won +9 more

Chemical mapping of the surface interactome of PIEZO1 identifies CADM1 as a modulator of channel inactivation

Proceedings of the National Academy of Sciences(2024)10.1073/pnas.2415934121

N/A

0DataRank · unranked

25 citations

Oleg Yarishkin, Adrienne E. Dubin, Jennifer M. Kefauver, Ryan A. Pak, Benjamin F. Cravatt +2 more

Covalent targeting of splicing in T cells

Cell chemical biology(2024)10.1016/j.chembiol.2024.10.010

N/A

0DataRank · unranked

16 citations

Hiroyuki Kojima, Nathalie Ropek, Charles David Warren, Tiffany L. Zhang, Simon J. Hogg +10 more

Chemical Proteomics–Guided Discovery of Covalent Ligands for Cancer Proteins

Annual Review of Cancer Biology(2024)10.1146/annurev-cancerbio-061421-041946

N/A

0DataRank · unranked

15 citations

Benjamin F. Cravatt, Xiaoyu Zhang

Exploiting the DCAF16–SPIN4 interaction to identify DCAF16 ligands for PROTAC development

RSC Medicinal Chemistry(2024)10.1039/d4md00681j

N/A

0DataRank · unranked

6 citations

Miguel Campos, Xiao‐Kang Jin, Fiona Y. Wang, Chenlu Zhang, Sara F. Dunne +3 more

SF3B1 thermostability as an assay for splicing inhibitor interactions

Journal of Biological Chemistry(2024)10.1016/j.jbc.2024.108135

N/A

0DataRank · unranked

5 citations

Guddeti Chandrashekar Reddy, Bruno Melillo, Benjamin F. Cravatt, Arun K. Ghosh, Melissa S. Jurica +1 more

Chemical probes for the identification of the molecular targets of honokiol

European Journal of Medicinal Chemistry(2024)10.1016/j.ejmech.2024.117102

N/A

0DataRank · unranked

4 citations

Ainoa Rueda‐Zubiaurre, D.M. Fernandez, Román Foronda, Christopher G. Parker, Benjamin F. Cravatt +3 more

Aspirin modulates generation of procoagulant phospholipids in cardiovascular disease, by regulating LPCAT3

Journal of Lipid Research(2024)10.1016/j.jlr.2024.100727

N/A

0DataRank · unranked

6 citations

Victoria J. Tyrrell, Ali A Hajeyah, Bethan Morgan, Daniela Costa, Yong Li +14 more

Redirecting the pioneering function of FOXA1 with covalent small molecules

bioRxiv (Cold Spring Harbor Laboratory)(2024)10.1101/2024.03.21.586158

N/A

0DataRank · unranked

10 citations

Yuxiang Zhang, Christopher J. Reinhardt, Nicole S. MacRae, Kristen E. DeMeester, Evert Njomen +6 more

Chemical tools to expand the ligandable proteome: diversity-oriented synthesis-based photoreactive stereoprobes

bioRxiv (Cold Spring Harbor Laboratory)(2024)10.1101/2024.02.27.582206

N/A

0DataRank · unranked

8 citations

David B. Konrad, Zher Yin Tan, Kimberly L. Carey, Jessica Y. Luo, Sang Joon Won +9 more

Enantiocontrolled Azetidine Library Synthesis via Strain-Release Functionalization of 1-Azabicyclobutanes

Journal of the American Chemical Society(2025)10.1021/jacs.5c07227

N/A

0DataRank · unranked

18 citations

Molhm Nassir, Hayden A. Sharma, Nathanyal J. Truax, Nicholas Raheja, Ty M. Thompson +5 more

Attenuating ABHD17 Isoforms Augments the S-acylation and Function of NOD2 and a Subset of Crohn’s Disease-associated NOD2 Variants

Cellular and Molecular Gastroenterology and Hepatology(2025)10.1016/j.jcmgh.2025.101491

N/A

0DataRank · unranked

10 citations

Noah R. Martin, Micah J. Niphakis, Benjamin F. Cravatt, Gregory D. Fairn, Charneal L. Dixon

Development of a novel 18F-labeled reversible-binding radioligand for imaging monoacylglycerol lipase with positron emission tomography

Acta Pharmaceutica Sinica B(2025)10.1016/j.apsb.2025.05.041

N/A

0DataRank · unranked

3 citations

Chunyu Zhao, Ahmad Chaudhary, Tim Ware, Richard Van, Yinlong Li +16 more

Intralysosomal Amyloidogenesis and Proximity Labeling by Cathepsin C

bioRxiv (Cold Spring Harbor Laboratory)(2025)10.64898/2025.12.23.696283

N/A

0DataRank · unranked

6 citations

Robert T. O’Neill, Idil Itir Demiralp, Seth Allen, Daniel Serwas, Hannah Siems +9 more

In vivo validation of the palmitoylation cycle as a therapeutic target in NRAS -mutant cancer

bioRxiv (Cold Spring Harbor Laboratory)(2025)10.1101/2025.03.20.644389

N/A

0DataRank · unranked

2 citations

Benjamin J. Huang, Timothy B. Ware, Christopher Boone, Michelle Tang, Julia Ybarra +25 more

Proteomic Ligandability Maps of Phosphorus(V) Stereoprobes Identify Covalent TLCD1 Inhibitors

bioRxiv (Cold Spring Harbor Laboratory)(2025)10.1101/2025.01.31.635883

N/A

0DataRank · unranked

1 citations

Michael Bielecki, Meredith A. Holm, Ty M. Thompson, Yue Yin, Jacob B. Cravatt +9 more

Erucamide regulates retinal neurovascular crosstalk

bioRxiv (Cold Spring Harbor Laboratory)(2025)10.1101/2025.09.02.673793

N/A

0DataRank · unranked

1 citations

Shreyosree Chatterjee, Qinglin Yang, Sanahan Vijayakumar, Daisuke Ogasawara, Sarah Giles +15 more

A chemical-genetic interaction between PAF1 and ENL/AF9 YEATS inhibition

bioRxiv (Cold Spring Harbor Laboratory)(2025)10.1101/2025.09.09.675200

N/A

0DataRank · unranked

0 citations

Leopold Garnar-Wortzel, D. Timothy Bishop, Rachel E. Hayward, Lauren M Hargis, James B. Shaum +5 more

A chemical-genetic interaction between PAF1 and ENL/AF9 YEATS inhibition

RSC Chemical Biology(2025)10.1039/d5cb00233h

N/A

0DataRank · unranked

0 citations

Leopold Garnar-Wortzel, Timothy Bishop, Rachel E. Hayward, Lauren Hargis, James B. Shaum +5 more

Mitochondrial ABHD11 inhibition drives sterol metabolism to modulate T-cell effector function

Nature Communications(2025)10.1038/s41467-025-65417-4

N/A

0DataRank · unranked

0 citations

Yasmin R Jenkins, Fernando M. Ponce-Garcia, Chloe Moscrop, Iain Perry, Matthew D. Hitchings +29 more

Covalent Targeting of Splicing in T Cells

bioRxiv (Cold Spring Harbor Laboratory)(2023)10.1101/2023.12.18.572199

N/A

0DataRank · unranked

5 citations

Hiroyuki Kojima, Nathalie Ropek, Charles David Warren, Tiffany L. Zhang, Simon J. Hogg +9 more

Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice

Nature Chemical Biology(2020)10.1038/s41589-020-0528-7

N/A

0DataRank · unranked

96 citations

Mohammed Ahmed Mustafa, Ozge Gunduz‐Cinar, Reşat Çınar, Gavin N. Petrie, Vasudev Kantae +34 more

AIG1 and ADTRP are endogenous hydrolases of fatty acid esters of hydroxy fatty acids (FAHFAs) in mice

Journal of Biological Chemistry(2020)10.1074/jbc.ra119.012145

N/A

0DataRank · unranked

47 citations

Bernard P. Kok, William H. Parsons, Justin Wang, Dan Tan, Cynthia J. Donaldson +11 more

Genetic disruption of N-RasG12D palmitoylation perturbs hematopoiesis and prevents myeloid transformation in mice

Blood(2020)10.1182/blood.2019003530

N/A

0DataRank · unranked

40 citations

Ari J. Firestone, Jarrett R. Remsberg, Benjamin J. Huang, Jasmine C. Wong, Amanda M. Long +8 more

Integrative X-ray Structure and Molecular Modeling for the Rationalization of Procaspase-8 Inhibitor Potency and Selectivity

ACS Chemical Biology(2020)10.1021/acschembio.0c00019

N/A

0DataRank · unranked

17 citations

Jérôme Eberhardt, Brianna Hill-Payne, Gonzalo E. González‐Páez, José O. Castellón, Benjamin F. Cravatt +4 more

Inhibition of monoacylglycerol lipase reduces nicotine reward in the conditioned place preference test in male mice

Neuropharmacology(2020)10.1016/j.neuropharm.2020.108170

N/A

0DataRank · unranked

12 citations

Lois S. Akinola, Joel E. Schlosburg, Aron H. Lichtman, Laura J. Sim‐Selley, Anu Mahadevan +3 more

Cell-Based Ligand Discovery for the ENL YEATS Domain

ACS Chemical Biology(2020)10.1021/acschembio.0c00124

N/A

0DataRank · unranked

38 citations

Natalia Milosevich, Emily Chen, Timothy Bishop, Justin Wang, Yuxiang Zhang +7 more

ABHD12 and LPCAT3 Interplay Regulates a Lyso-phosphatidylserine-C20:4 Phosphatidylserine Lipid Network Implicated in Neurological Disease

Biochemistry(2020)10.1021/acs.biochem.0c00292

N/A

0DataRank · unranked

35 citations

Alex Reed, Daisuke Ogasawara, Olesya A. Ulanovskaya, Amanda J. Roberts, Carlos Aguirre +9 more

Physical and Functional Analysis of the Putative Rpn13 Inhibitor RA190

Cell chemical biology(2020)10.1016/j.chembiol.2020.08.007

N/A

0DataRank · unranked

28 citations

Daniel Abegg, Ekaterina V. Vinogradova, Junichiro Takaya, Hongchan An, Scott Simanski +4 more

Chemical inhibition of ENL/AF9 YEATS domains in acute leukemia

bioRxiv (Cold Spring Harbor Laboratory)(2020)10.1101/2020.12.01.406694

N/A

0DataRank · unranked

5 citations

Timothy Bishop, Seiya Kitamura, Natalia Milosevich, Joshua N. Asiaban, Xiaoyu Zhang +13 more

ABHD17 enzymes regulate dynamic plasma membrane palmitoylation and N-Ras-dependent cancer growth

bioRxiv (Cold Spring Harbor Laboratory)(2020)10.1101/2020.05.21.108316

N/A

0DataRank · unranked

2 citations

Radu M. Suciu, Noemi A. Zambetti, Thomas W. Hanigan, Ari J. Firestone, Anagha Inguva Sheth +12 more

Paracrine Induction of HIF by Glutamate in Breast Cancer: EglN1 Senses Cysteine

UNC Libraries(2020)10.17615/emqc-jb75

N/A

0DataRank · unranked

0 citations

Kimberly J. Briggs, Agnieszka K. Witkiewicz, Shugeng Cao, Benjamin F. Cravatt, Keriann M. Backus +9 more

A proteome-wide atlas of lysine-reactive chemistry

Nature Chemistry(2021)10.1038/s41557-021-00765-4

N/A

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