Daniel A. Harki

Biochemistry, Genetics and Molecular BiologyMedicineImmunology and Microbiology

Pilot corpus only

This score is computed over theSindex pilot corpus and does not cover the full scientific literature. Scores are relative to papers we have ingested — papers, authors, and institutions outside the pilot are not represented. Methodology.

Top 100%percentile

0Author DataRank

Indexed papers

0in pilot corpus

datarank_citation_only_1hop_v6· scope data_onlyMethodology

Papers

Driven by 29 papers. Top paper: “Selective N‐Terminal BET Bromodomain Inhibitors by Targeting Non‐Conserved Residues and Structured Water Displacement**”.

Selective N‐Terminal BET Bromodomain Inhibitors by Targeting Non‐Conserved Residues and Structured Water Displacement**

Angewandte Chemie International Edition(2020)10.1002/anie.202008625

N/A

0.574DataRank · unranked

45 citations

Anand Divakaran, Anil K. Pandey, Jorden A. Johnson, Huda Zahid, Zachariah J. Hoell +6 more

Development of an N-Terminal BRD4 Bromodomain-Targeted Degrader

ChemRxiv(2021)10.26434/chemrxiv-2021-zvq4t

N/A

0.104DataRank · unranked

1 citations

Huda Zahid, Wenwei Lin, Taosheng Chen, Daniel A. Harki, William C. K. Pomerantz +1 more

Induced copy-back RNA synthesis as a novel therapeutic mechanism against RNA viruses

bioRxiv (Cold Spring Harbor Laboratory)(2020)10.1101/2020.02.12.946558

N/A

0DataRank · unranked

8 citations

Andrew Woodman, Kuo-Ming Lee, Ibrahim M. Moustafa, Fiona Fitzgerald, Peng-Nien Huang +9 more

4-Methyl-1,2,3-Triazoles as N-Acetyl-Lysine Mimics Afford Potent BET Bromodomain Inhibitors with Improved Selectivity

Journal of Medicinal Chemistry(2021)10.1021/acs.jmedchem.1c00933

N/A

0DataRank · unranked

36 citations

Angela S. Carlson, Mary A. Schleiff, Anand Divakaran, Jorden A. Johnson, Caroline R. Buchholz +9 more

Induced intra- and intermolecular template switching as a therapeutic mechanism against RNA viruses

Molecular Cell(2021)10.1016/j.molcel.2021.10.003

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0DataRank · unranked

24 citations

Andrew Woodman, Djoshkun Shengjuler, Thomas Vallet, Kuo-Ming Lee, Louis Kuijpers +12 more

An efficient synthesis of RNA containing GS-441524: the nucleoside precursor of remdesivir

RSC Advances(2021)10.1039/d1ra06589k

N/A

0DataRank · unranked

4 citations

Samantha A. Kennelly, Deborah J. Rodriguez, Daniel A. Harki, Ramkumar Moorthy

Function‐Oriented and Modular (+/−)‐cis‐Pseudoguaianolide Synthesis: Discovery of New Nrf2 Activators and NF‐κB Inhibitors

Chemistry - A European Journal(2021)10.1002/chem.202100038

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0DataRank · unranked

7 citations

Ranjala Ratnayake, Henry A. M. Schares, Katherine F. M. Jones, Emily Bevan–Smith, Hendrik Luesch +3 more

Gain-of-Signal Assays for Probing Inhibition of SARS-CoV-2 M pro /3CL pro in Living Cells

mBio(2022)10.1128/mbio.00784-22

N/A

0DataRank · unranked

39 citations

Morgan A. Esler, Yuka Otsuka, Jordan T. Becker, Sofia N. Moraes, Constance B. Anderson +12 more

Interfering with nucleotide excision by the coronavirus 3′-to-5′ exoribonuclease

Nucleic Acids Research(2022)10.1093/nar/gkac1177

N/A

0DataRank · unranked

21 citations

Mohamad S. Sotoudegan, Pankaj Srivastava, Thomas K. Anderson, Ibrahim M. Moustafa, Kellan T. Passow +9 more

SARS-CoV-2 nsp14 Exoribonuclease Removes the Natural Antiviral 3′-Deoxy-3′,4′-didehydro-cytidine Nucleotide from RNA

Viruses(2022)10.3390/v14081790

N/A

0DataRank · unranked

16 citations

Kellan T. Passow, Daniel A. Harki, Hideki Aihara, Nicholas H. Moeller

A synthetic covalent ligand of the C/EBPβ transactivation domain inhibits acute myeloid leukemia cells

Cancer Letters(2022)10.1016/j.canlet.2022.01.024

N/A

0DataRank · unranked

11 citations

Maria V. Yusenko, Daria Frank, Ramkumar Moorthy, John C. Widen, Wolfgang Dörner +4 more

Targeting N-Myc in Neuroblastoma with Selective Aurora Kinase A Degraders

bioRxiv (Cold Spring Harbor Laboratory)(2022)10.1101/2022.04.09.487756

N/A

0DataRank · unranked

5 citations

Ramkumar Moorthy, Özlem Demir, Zachary D. Baker, Jordan A. Naumann, Katherine F. M. Jones +10 more

Development of allosteric, selective cyclin-dependent kinase 2 (CDK2) inhibitors that are negatively cooperative with cyclin binding and show potential as contraceptive agents

bioRxiv (Cold Spring Harbor Laboratory)(2022)10.1101/2022.06.30.497818

N/A

0DataRank · unranked

4 citations

Jian Tang, Emily Roberts, Sornakala Ganeshkumar, Luxin Sun, Nan Wang +12 more

Interfering with nucleotide excision by the coronavirus 3’-to-5’ exoribonuclease

bioRxiv (Cold Spring Harbor Laboratory)(2022)10.1101/2022.08.11.503614

N/A

0DataRank · unranked

0 citations

Mohamad S. Sotoudegan, Thomas K. Anderson, Ibrahim M. Moustafa, Kellan T. Passow, Samantha A. Kennelly +8 more

A Chemical Strategy for Intracellular Arming of an Endogenous Broad-Spectrum Antiviral Nucleotide

Figshare(2022)10.17615/hy4j-3r92

N/A

0DataRank · unranked

0 citations

Anoop Narayanan, Nicole M. Antczak, Craig E. Cameron, Daniel A. Harki, Joyce Jose +6 more

Development of allosteric and selective CDK2 inhibitors for contraception with negative cooperativity to cyclin binding

Nature Communications(2023)10.1038/s41467-023-38732-x

N/A

0DataRank · unranked

48 citations

Luxin Sun, Jian Tang, Emily Roberts, Sornakala Ganeshkumar, Nan Wang +13 more

4-Isocyanoindole-2ʹ-deoxyribonucleoside (4ICIN): An isomorphic indole nucleoside suitable for inverse electron demand Diels-Alder reactions

Tetrahedron Letters(2023)10.1016/j.tetlet.2023.154807

N/A

0DataRank · unranked

5 citations

Daniel A. Harki, Kellan T. Passow

Fragment-Based NMR Screening of the BPTF PHD Finger Methyl Lysine Reader Leads to the First Small-Molecule Inhibitors

ACS Medicinal Chemistry Letters(2023)10.1021/acsmedchemlett.3c00343

N/A

0DataRank · unranked

5 citations

Molly Sneddon, Joseph E. McPherson, Sourav Das, Clifford T. Gee, Michael J. Grillo +7 more

Development of Allosteric NIK Ligands from Fragment-Based NMR Screening

ACS Medicinal Chemistry Letters(2023)10.1021/acsmedchemlett.3c00429

N/A

0DataRank · unranked

5 citations

Michael J. Grillo, Daniel A. Harki, Jared J. Anderson

Synthesis and photophysical characterization of fluorescent indole nucleoside analogues

RSC Advances(2023)10.1039/d3ra03457g

N/A

0DataRank · unranked

4 citations

Kellan T. Passow, Daniel A. Harki, Jacob M. Sawyer

APOBEC3A Catalytic Inactivity Mutation Induces Tertiary Structure Destabilization

ACS Medicinal Chemistry Letters(2023)10.1021/acsmedchemlett.2c00517

N/A

0DataRank · unranked

4 citations

Mohamed Shehata, Michael A. Carpenter, Rommie E. Amaro, Daniel A. Harki, Katherine F. M. Jones

Fragment-Based NMR Screening of the BPTF PHD Finger Methyl Lysine Reader Leads to the First Small Molecule Inhibitors

ChemRxiv(2023)10.26434/chemrxiv-2023-8t7wn

N/A

0DataRank · unranked

1 citations

Molly Sneddon, Joseph McPherson, Sourav Das, Clifford T. Gee, Michael A. Grillo +7 more

Interfering with nucleotide excision by the coronavirus 3′-to-5′ exoribonuclease

UNC Libraries(2023)10.17615/k1hp-as05

N/A

0DataRank · unranked

0 citations

Thomas K. Anderson, Joy Y. Feng, Pankaj Srivastava, Rukesh Chinthapatla, Kellan T. Passow +9 more

A compact stem-loop DNA aptamer targets a uracil-binding pocket in the SARS-CoV-2 nucleocapsid RNA-binding domain

Nucleic Acids Research(2024)10.1093/nar/gkae874

N/A

0DataRank · unranked

18 citations

Christopher Belica, Joseph A. Rollie, William L. Brown, Seyed Arad Moghadasi, Ke Shi +4 more

SARS-CoV-2 Mpro inhibitor identification using a cellular gain-of-signal assay for high-throughput screening

SLAS DISCOVERY(2024)10.1016/j.slasd.2024.100181

N/A

0DataRank · unranked

6 citations

Jyoti Vishwakarma, Seyed Arad Moghadasi, Yuka Otsuka, Justin Shumate, Ashley Cuell +14 more

Development of Allosteric Small Molecule APOBEC3B Inhibitors from In Silico Screening

bioRxiv (Cold Spring Harbor Laboratory)(2024)10.1101/2024.04.25.591187

N/A

0DataRank · unranked

0 citations

Özlem Demir, Mackenzie K. Wyllie, Michael J. Grillo, Clare K. Morris, Sophia P. Hirakis +6 more

Targeting N-Myc in neuroblastoma with selective Aurora kinase A degraders

Cell chemical biology(2025)10.1016/j.chembiol.2024.12.006

N/A

0DataRank · unranked

23 citations

Ramkumar Moorthy, Laura Hirsch, Özlem Demir, Zachary D. Baker, Jordan A. Naumann +12 more

Identification of a novel allosteric binding site on the catalytic domain of NF-κB inducing kinase (NIK)

RSC Medicinal Chemistry(2025)10.1039/d4md00963k

N/A

0DataRank · unranked

1 citations

Daniel A. Harki, Jared J. Anderson

Selective N‐Terminal BET Bromodomain Inhibitors by Targeting Non‐Conserved Residues and Structured Water Displacement**

Angewandte Chemie(2020)10.1002/ange.202008625

N/A

0DataRank · unranked

2 citations

Anand Divakaran, Anil K. Pandey, Jorden A. Johnson, Huda Zahid, Zachariah J. Hoell +6 more