Terrence R. Burke

Also affiliated with Frederick National Laboratory for Cancer Research, National Cancer Institute, Center for Cancer Research

Biochemistry, Genetics and Molecular BiologyMedicineImmunology and Microbiology

Pilot corpus only

This score is computed over theSindex pilot corpus and does not cover the full scientific literature. Scores are relative to papers we have ingested — papers, authors, and institutions outside the pilot are not represented. Methodology.

Top 100%percentile

0Author DataRank

Indexed papers

0in pilot corpus

datarank_citation_only_1hop_v6· scope data_onlyMethodology

Papers

Driven by 29 papers. Top paper: “Mechanisms of HIV-1 integrase resistance to dolutegravir and potent inhibition of drug-resistant variants”.

Mechanisms of HIV-1 integrase resistance to dolutegravir and potent inhibition of drug-resistant variants

Science Advances(2023)10.1126/sciadv.adg5953

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0.843DataRank · unranked

38 citations

Dario Oliveira Passos, Zelin Shan, Steven J. Smith, Qinfang Sun, Avik Biswas +14 more

Small molecule microarray identifies inhibitors of tyrosyl-DNA phosphodiesterase 1 that simultaneously access the catalytic pocket and two substrate binding sites

Chemical Science(2021)10.1039/d0sc05411a

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0.529DataRank · unranked

33 citations

Evgeny Kiselev, G.T. Lountos, Wenjie Wang, Joseph E. Tropea, D. Needle +6 more

Structural basis for the inhibition of HTLV-1 integration inferred from cryo-EM deltaretroviral intasome structures

Nature Communications(2021)10.1038/s41467-021-25284-1

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0.457DataRank · unranked

20 citations

Teresa Vanzo, Xue Zhi Zhao, Steven J. Smith, Allison Ballandras-Colas, Nora Cronin +6 more

Targeted sulfur(VI) fluoride exchange-mediated covalent modification of a tyrosine residue in the catalytic pocket of tyrosyl-DNA phosphodiesterase 1

Communications Chemistry(2024)10.1038/s42004-024-01298-w

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0.312DataRank · unranked

7 citations

I Barakat, G.T. Lountos, Wenjie Wang, Keli Agama, Md Rasel Al Mahmud +5 more

Comparative Analyses of Antiviral Potencies of Second-Generation Integrase Strand Transfer Inhibitors (INSTIs) and the Developmental Compound 4d Against a Panel of Integrase Quadruple Mutants

Viruses(2025)10.3390/v17010121

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0.165DataRank · unranked

2 citations

Xue Zhi Zhao, Stephen H. Hughes, Terrence R. Burke, Steven J. Smith

A new genre of fluorescence recovery assay to evaluate polo-like kinase 1 ATP-competitive inhibitors

Analytical Methods(2020)10.1039/d0ay01223h

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0DataRank · unranked

3 citations

David Hymel, Terrence R. Burke, Kohei Tsuji

Application of Post Solid-Phase Oxime Ligation to Fine-Tune Peptide–Protein Interactions

Molecules(2020)10.3390/molecules25122807

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0DataRank · unranked

1 citations

Fa Liu, Terrence R. Burke, Xue Zhi Zhao

Integrase Strand Transfer Inhibitors Are Effective Anti-HIV Drugs

Viruses(2021)10.3390/v13020205

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0DataRank · unranked

104 citations

Xue Zhi Zhao, Dario Oliveira Passos, Dmitry Lyumkis, Terrence R. Burke, Stephen H. Hughes +1 more

Design and synthesis of a new orthogonally protected glutamic acid analog and its use in the preparation of high affinity polo-like kinase 1 polo-box domain – binding peptide macrocycles

Organic & Biomolecular Chemistry(2021)10.1039/d1ob01120k

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0DataRank · unranked

10 citations

Kohei Tsuji, Robert A. Grant, Ramesh Chingle, Dominique L. Kunciw, Michael B Yaffe +2 more

Development of ultra-high affinity bivalent ligands targeting the polo-like kinase 1

RSC Chemical Biology(2022)10.1039/d2cb00153e

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0DataRank · unranked

12 citations

David Hymel, Buyong Ma, Hirokazu Tamamura, Ruth Nussinov, Terrence R. Burke +1 more

Phosphonic acid-containing inhibitors of tyrosyl-DNA phosphodiesterase 1

Frontiers in Chemistry(2022)10.3389/fchem.2022.910953

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0DataRank · unranked

8 citations

Wenjie Wang, G.T. Lountos, Joseph E. Tropea, D. Needle, Yves Pommier +2 more

Mechanisms of HIV-1 Integrase Resistance to Dolutegravir and Potent Inhibition of Drug Resistant Variants

bioRxiv (Cold Spring Harbor Laboratory)(2022)10.1101/2022.12.04.519057

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0DataRank · unranked

3 citations

Dario Oliveira Passos, Zelin Shan, Steven J. Smith, Qinfang Sun, Avik Biswas +12 more

Synthetic Approaches to a Key Pyridone-carboxylic Acid Precursor Common to the HIV-1 Integrase Strand Transfer Inhibitors Dolutegravir, Bictegravir, and Cabotegravir

Organic Process Research & Development(2023)10.1021/acs.oprd.3c00063

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0DataRank · unranked

8 citations

Terrence R. Burke, Pankaj S. Mahajan

Identification of multidentate tyrosyl-DNA phosphodiesterase 1 (TDP1) inhibitors that simultaneously access the DNA, protein and catalytic-binding sites by oxime diversification

RSC Chemical Biology(2023)10.1039/d2cb00230b

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0DataRank · unranked

10 citations

Wenjie Wang, G.T. Lountos, Evgeny Kiselev, Joseph E. Tropea, D. Needle +3 more

A Practical Approach to Bicyclic Carbamoyl Pyridones with Application to the Synthesis of HIV-1 Integrase Strand Transfer Inhibitors

Molecules(2023)10.3390/molecules28031428

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0DataRank · unranked

5 citations

Steven J. Smith, Stephen H. Hughes, Xue Zhi Zhao, Terrence R. Burke, Pankaj S. Mahajan

Examination of aminophenol-containing compounds designed as antiproliferative agents and potential atypical retinoids

Bioorganic & Medicinal Chemistry(2023)10.1016/j.bmc.2023.117214

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0DataRank · unranked

4 citations

Masahiko Imai, Sarah E. Altman, Daisuke Saito, Noriko Takahashi, Terrence R. Burke +1 more

Affinity enhancement of polo-like kinase 1 polo box domain-binding ligands by a bivalent approach using a covalent kinase-binding component

RSC Chemical Biology(2024)10.1039/d4cb00031e

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0DataRank · unranked

5 citations

Hirokazu Tamamura, Terrence R. Burke, Kohei Tsuji

N-Substituted Bicyclic Carbamoyl Pyridones: Integrase Strand Transfer Inhibitors that Potently Inhibit Drug-Resistant HIV-1 Integrase Mutants

ACS Infectious Diseases(2024)10.1021/acsinfecdis.3c00525

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0DataRank · unranked

4 citations

Steven J. Smith, Min Li, Robert Craigie, Stephen H. Hughes, Xue Zhi Zhao +2 more

Application of a Fluorescence Recovery-Based Polo-Like Kinase 1 Binding Assay to Polo-Like Kinase 2 and Polo-Like Kinase 3

Biological and Pharmaceutical Bulletin(2024)10.1248/bpb.b24-00189

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0DataRank · unranked

3 citations

Hirokazu Tamamura, Terrence R. Burke, Kohei Tsuji

Fine-tuning probes for fluorescence polarization binding assays of bivalent ligands against polo-like kinase 1 using full-length protein

Bioorganic & Medicinal Chemistry(2024)10.1016/j.bmc.2024.118055

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0DataRank · unranked

2 citations

Hirokazu Tamamura, Terrence R. Burke, Kohei Tsuji

Enhancing precision in colorectal cancer surgery: development of an LGR5-targeting RSPO1 peptide mimetic as a contrast agent for intraoperative fluorescence molecular imaging

Cell Cycle(2024)10.1080/15384101.2024.2364578

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0DataRank · unranked

1 citations

Patrícia Ribeiro, Ramesh Chingle, Thomas Rohwetter, Nikita Gupta, George Avetian +11 more

Application of a bivalent “click” approach to target tyrosyl-DNA phosphodiesterase 1 (TDP1)

RSC Medicinal Chemistry(2025)10.1039/d4md00824c

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0DataRank · unranked

4 citations

Wenjie Wang, Md Rasel Al Mahmud, Keli Agama, Yves Pommier, Terrence R. Burke +1 more

Pi–pi stacking interactions with viral DNA contribute to the potency of naphthyridine-based HIV-1 integrase inhibitors

NAR Molecular Medicine(2025)10.1093/narmme/ugaf039

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0DataRank · unranked

2 citations

Min Li, Steven J. Smith, Arvin Karbasi, Indrani Choudhuri, Tao Jing +4 more

Structural basis for strand-transfer inhibitor binding to HIV intasomes

Science(2020)10.1126/science.aay8015

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0DataRank · unranked

111 citations

Min Li, I.K. Jozwik, Xue Zhi Zhao, Diogo Santos‐Martins, Renbin Yang +8 more

Potent β-lactam-based tyrosyl-DNA phosphodiesterase 1 inhibitors identified by a virtual screen

Scientific Reports(2025)10.1038/s41598-025-12503-8

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0DataRank · unranked

1 citations

Wenjie Wang, Kiall F. Suazo, Md Rasel Al Mahmud, Keli Agama, G.T. Lountos +4 more

Uncoupling the Folding-Function Paradigm of Lytic Peptides to Deliver Impermeable Inhibitors of Intracellular Protein–Protein Interactions

Journal of the American Chemical Society(2020)10.1021/jacs.0c07921

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0DataRank · unranked

21 citations

Kohei Tsuji, Rachel P. M. Abrams, Terrence R. Burke, Joel P. Schneider, Stephen E. Miller

Chemically Programmable and Switchable CAR‐T Therapy

Angewandte Chemie International Edition(2020)10.1002/anie.202005432

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0DataRank · unranked

44 citations

Kohei Tsuji, David Hymel, Terrence R. Burke, Michael Hudecek, Christoph Rader +2 more

HIV-1 Integrase Inhibitors That Are Active against Drug-Resistant Integrase Mutants

Antimicrobial Agents and Chemotherapy(2020)10.1128/aac.00611-20

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0DataRank · unranked

32 citations

Xue Zhi Zhao, Dario Oliveira Passos, Dmitry Lyumkis, Terrence R. Burke, Stephen H. Hughes +1 more

Chemically Programmable and Switchable CAR‐T Therapy

Angewandte Chemie(2020)10.1002/ange.202005432

N/A

0DataRank · unranked

7 citations

Kohei Tsuji, David Hymel, Terrence R. Burke, Michael Hudecek, Christoph Rader +2 more