Wayne E. Childers

Biochemistry, Genetics and Molecular BiologyChemistryNeuroscience

Pilot corpus only

This score is computed over theSindex pilot corpus and does not cover the full scientific literature. Scores are relative to papers we have ingested — papers, authors, and institutions outside the pilot are not represented. Methodology.

Top 100%percentile

0Author DataRank

Indexed papers

1in pilot corpus

datarank_citation_only_1hop_v6· scope data_onlyMethodology

Why this DataRank?

An author's DataRank is the sum of the DataRanks of all 1 indexed paper attributed to them. A prolific author with many moderate-impact papers can outrank one with a single high-impact paper.

Author scores recompute whenever paper DataRanks are refreshed, so this number lags the underlying paper scores by at most one batch run.

Read the full methodology →

Papers

Driven by 21 papers. Top paper: “The Resurrection of Phenotypic Drug Discovery”.

The Resurrection of Phenotypic Drug Discovery

ACS Medicinal Chemistry Letters(2020)10.1021/acsmedchemlett.0c00006

N/A

0.578DataRank · unranked

46 citations

Khaled M. Elokely, Magid Abou‐Gharbia, Wayne E. Childers

Structure–Activity Relationship of a Pyrrole Based Series of PfPKG Inhibitors as Anti-Malarials

Journal of Medicinal Chemistry(2024)10.1021/acs.jmedchem.3c01795

N/A

0.406DataRank · unranked

14 citations

Kutub Ashraf, Melvin Delvillar, Tyler Eck, Raheel Fondekar, Edward B. Miller +15 more

Neuroinflammation and Neurometabolomic Profiling in Fentanyl Overdose Mouse Model Treated with Novel β-Lactam, MC-100093, and Ceftriaxone

Toxics(2024)10.3390/toxics12080604

N/A

0.345DataRank · unranked

9 citations

Fawaz Alasmari, Shakir D. AlSharari, Abdullah F. Alasmari, Nemat Ali, Syed Rizwan Ahamad +8 more

Effects of novel beta-lactam, MC-100093, and ceftriaxone on astrocytic glutamate transporters and neuroinflammatory factors in nucleus accumbens of C57BL/6 mice exposed to escalated doses of morphine

Saudi Pharmaceutical Journal(2024)10.1016/j.jsps.2024.102108

N/A

0.312DataRank · unranked

7 citations

Ghadeer M.S. Swiss, Fatin A. Alrashedi, Kholoud A. Baeshen, Sultan A. Alshammari, Shakir D. AlSharari +8 more

DYRK1A inhibition results in MYC and ERK activation rendering KMT2A-R acute lymphoblastic leukemia cells sensitive to BCL2 inhibition

Leukemia(2025)10.1038/s41375-025-02575-w

N/A

0.219DataRank · unranked

3 citations

Gerald Wertheim, Shikha Gaur, John Chukinas, Joseph P. Loftus, Sung June Lee +15 more

First Optimization of Novel, Potent, Selective PDE11A4 Inhibitors for Age-Related Cognitive Decline

Journal of Medicinal Chemistry(2023)10.1021/acs.jmedchem.3c01088

N/A

0DataRank · unranked

9 citations

Mariana Lozano Gonzalez, Sreedhar R. Tummalapalli, Jeremy Eberhard, Judy Ly, Charles S. Hoffman +6 more

Discovery of a small-molecule inhibitor that traps Polθ on DNA and synergizes with PARP inhibitors

Nature Communications(2024)10.1038/s41467-024-46593-1

N/A

0DataRank · unranked

47 citations

Mrityunjay Tyagi, Leonid Minakhin, Gurushankar Chandramouly, Taylor Tredinnick, Mercy Ramanjulu +18 more

Effects of a Novel Beta Lactam Compound, MC-100093, on the Expression of Glutamate Transporters/Receptors and Ethanol Drinking Behavior of Alcohol-Preferring Rats

Journal of Pharmacology and Experimental Therapeutics(2022)10.1124/jpet.122.001147

N/A

0DataRank · unranked

17 citations

Woonyen Wong, Magid Abou‐Gharbia, Wayne E. Childers, Edward Melenski, Richard L. Bell +2 more

Effects of novel GLT-1 modulator, MC-100093, on neuroinflammatory and neurotrophic biomarkers in mesocorticolimbic brain regions of male alcohol preferring rats exposed chronically to ethanol

Brain Research Bulletin(2024)10.1016/j.brainresbull.2024.110935

N/A

0DataRank · unranked

9 citations

Ahmed Alotaibi, Woonyen Wong, Magid Abou‐Gharbia, Wayne E. Childers, Youssef Sari +1 more

Discovery of imidazole-based inhibitors of P. falciparum cGMP-dependent protein kinase

bioRxiv (Cold Spring Harbor Laboratory)(2021)10.1101/2021.11.05.467463

N/A

0DataRank · unranked

0 citations

Mariana Laureano de Souza, Mariana Lozano Gonzalez, Shams Ul Mahmood, Tyler Eck, Tamara Kreiss +11 more

MC-100093, a Novel β-Lactam Glutamate Transporter-1 Enhancer Devoid of Antimicrobial Properties, Attenuates Cocaine Relapse in Rats

Journal of Pharmacology and Experimental Therapeutics(2021)10.1124/jpet.121.000532

N/A

0DataRank · unranked

20 citations

Lizhen Wu, Jeffrey Rothstein, Svetlana Vidensky, John Gordon, Mercy Ramanjulu +5 more

Effects of MC-100093 on Ethanol Drinking and the Expression of Astrocytic Glutamate Transporters in the Mesocorticolimbic Brain Regions of Male and Female Alcohol-Preferring Rats

Neuroscience(2024)10.1016/j.neuroscience.2024.06.017

N/A

0DataRank · unranked

7 citations

Shelby Travaglianti, Woonyen Wong, Magid Abou‐Gharbia, Wayne E. Childers, Youssef Sari +1 more

MC180295 is a highly potent and selective CDK9 inhibitor with preclinical in vitro and in vivo efficacy in cancer

Clinical Epigenetics(2024)10.1186/s13148-023-01617-3

N/A

0DataRank · unranked

5 citations

Chen Huang, John Gordon, Sijia Yu, George Morton, Wayne E. Childers +5 more

First Demonstration of In Vivo PDE11A4 Target Engagement for Potential Treatment of Age-Related Memory Disorders

Journal of Medicinal Chemistry(2024)10.1021/acs.jmedchem.4c01794

N/A

0DataRank · unranked

4 citations

Jeremy Eberhard, Charles S. Hoffman, Dennis Colussi, John Gordon, Wayne E. Childers +5 more

Novel inhibitors of acute, axonal DLK palmitoylation are neuroprotective and avoid the deleterious side effects of cell-wide DLK inhibition

bioRxiv (Cold Spring Harbor Laboratory)(2024)10.1101/2024.04.19.590310

N/A

0DataRank · unranked

7 citations

Hey‐Kyeong Jeong, Jingwen Niu, Sabrina Holland, Brittany N. Rotanz, John Gordon +4 more

Correction to “Structure–Activity Relationship of a Pyrrole Based Series of PfPKG Inhibitors as Anti-Malarials”

Journal of Medicinal Chemistry(2024)10.1021/acs.jmedchem.4c01411

N/A

0DataRank · unranked

1 citations

Kutub Ashraf, Melvin Delvillar, Tyler Eck, Raheel Fondekar, Edward B. Miller +15 more

Inhibiting acute, axonal DLK palmitoylation is neuroprotective and avoids deleterious effects of cell-wide DLK inhibition

Nature Communications(2025)10.1038/s41467-025-58036-6

N/A

0DataRank · unranked

6 citations

Hey‐Kyeong Jeong, Jingwen Niu, Sabrina Holland, Brittany N. Rotanz, John Gordon +4 more

Mechanistic studies on pH-permeability relationships: Impact of the membrane polar headgroup region on pKa

International Journal of Pharmaceutics(2025)10.1016/j.ijpharm.2025.125383

N/A

0DataRank · unranked

4 citations

Irfan Khan, Mercy Ramanjulu, Paul Anthony, Wayne E. Childers, Swati Nagar +2 more

Differential Modulation of Glutamate Transporter‐1 by Cocaine and Oxycodone and the Efficacy of MC‐100093 to Reduce Reinstatement of Self‐Administration

Brain and Behavior(2025)10.1002/brb3.70616

N/A

0DataRank · unranked

1 citations

Yanaira Alonso‐Caraballo, Britta Hornback, Angel Robert, Megan A. Brickner, Manuel Esguerra +4 more

Liver Metabolomics and Inflammatory Profiles in Mouse Model of Fentanyl Overdose Treated with Beta-Lactams

Metabolites(2023)10.3390/metabo13080965

N/A

0DataRank · unranked

14 citations

Mohammed Alasmari, Mohammed A. Assiri, Mohammed Alswayyed, Syed Rizwan Ahamad, Abdulrahman I. Alhumaydhi +8 more

Discovery of novel potent, cell-permeable inhibitors of P. falciparum cGMP-dependent protein kinase

bioRxiv (Cold Spring Harbor Laboratory)(2021)10.1101/2021.08.24.457553

N/A

0DataRank · unranked

0 citations

Mariana Lozano Gonzalez, Shams Ul Mahmood, Tyler Eck, Tamara Kreiss, Mariana Laureano de Souza +11 more