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Focused structure-activity relationship profiling around the 2-phenylindole scaffold of a cannabinoid type-1 receptor agonist-positive allosteric modulator: site-III aromatic-ring congeners with enhanced activity and solubility

Bioorganic & Medicinal Chemistry(2020)10.1016/j.bmc.2020.115727Source: DataRank Database

Focused structure-activity relationship profiling around the 2-phenylindole scaffold of a cannabinoid type-1 receptor agonist-positive allosteric modulator: site-III aromatic-ring congeners with enhanced activity and solubility is a research paper published in Bioorganic & Medicinal Chemistry (2020). On theSindex it has a DataRank of 0. It has been cited 9 times.

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Open Access9 citations

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›Methodology & internals

datarank_citation_only_1hop_v6· scope data_onlyMethodology

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Enrichment:Funding (2 grants)Impact (FWCI 0.37)OA: greenTopics (47)IDs (PubMed, OpenAlex)SDGs (1)

FAIR Checklist

Context only (not used in score)

Findable (1/2)

Has DOI

Accessible (1/2)

Open Access

Interoperable (0/2)

Reusable (0/3)

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Authors (4)

Pushkar M. Kulkarni ORCID,David R. Janero ORCID,Ganesh A. Thakur,Peter C. Schaffer

Live enrichment

PubMed:33065437 OpenAlex:https://openalex.org/W3082718442

National Institutes of Health

Grant: EY024727

National Institutes of Health

Grant: EY024717

FWCI

0.37

Citation Percentile

0.6%

Citation Trend

2021

2022

2023

2024

2025

2026

greenLicense: https://www.elsevier.com/legal/tdmrep-license

repositoryhttps://doi.org/10.7270/q2bk1h05

publisherhttps://api.elsevier.com/content/article/PII:S0968089620305575?httpAccept=text/xml

publisherhttps://api.elsevier.com/content/article/PII:S0968089620305575?httpAccept=text/plain

journalhttps://doi.org/10.1016/j.bmc.2020.115727

Fields of Study

Pharmacological Receptor Mechanisms and EffectsCannabis and Cannabinoid ResearchReceptor Mechanisms and SignalingAllosteric RegulationAllosteric SiteCannabinoid Receptor AgonistsHumansIndolesKineticsMolecular Docking SimulationReceptor, Cannabinoid, CB1SolubilityStructure-Activity Relationshipbeta-Arrestins

MeSH Terms

beta-ArrestinsAllosteric RegulationAllosteric SiteHumansIndolesKineticsSolubilityStructure-Activity RelationshipReceptor, Cannabinoid, CB1Molecular Docking SimulationCannabinoid Receptor Agonists

Keywords

ChemistryAllosteric regulationStructure–activity relationshipCannabinoidAllosteric modulatorLead compoundAgonistStereochemistryCombinatorial chemistryIntrinsic activitySmall moleculeDrug discoverySolubilityReceptorIn vitroBiochemistryOrganic chemistryPositive Allosteric ModulatorFunctional SelectivityCannabinoid Type-1 ReceptorPhysiochemical Properties2-Phenylindole

Sustainable Development Goals

SDG 0: Clean water and sanitation