Retheesh S. Thankan

Pilot corpus only

This score is computed over theSindex pilot corpus and does not cover the full scientific literature. Scores are relative to papers we have ingested — papers, authors, and institutions outside the pilot are not represented. Methodology.

Top 100%percentile

0Author DataRank

Indexed papers

0in pilot corpus

datarank_citation_only_1hop_v6· scope data_onlyMethodology

Papers

Driven by 7 papers. Top paper: “Transcriptome profiling reveals that VNPP433‐3β, the lead next‐generation galeterone analog inhibits prostate cancer stem cells by downregulating epithelial–mesenchymal transition and stem cell markers”.

Transcriptome profiling reveals that VNPP433‐3β, the lead next‐generation galeterone analog inhibits prostate cancer stem cells by downregulating epithelial–mesenchymal transition and stem cell markers

Molecular Carcinogenesis(2022)10.1002/mc.23406

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0DataRank · unranked

31 citations

Retheesh S. Thankan, Puranik Purushottamachar, Weiliang Huang, Maureen A. Kane, Yuji Zhang +4 more

Novel AR/AR-V7 and Mnk1/2 Degrader, VNPP433-3β: Molecular Mechanisms of Action and Efficacy in AR-Overexpressing Castration Resistant Prostate Cancer In Vitro and In Vivo Models

Cells(2022)10.3390/cells11172699

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0DataRank · unranked

15 citations

Retheesh S. Thankan, Puranik Purushottamachar, Weiliang Huang, Maureen A. Kane, Yuji Zhang +4 more

Large-scale synthesis of galeterone and lead next generation galeterone analog VNPP433-3β

Steroids(2022)10.1016/j.steroids.2022.109062

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0DataRank · unranked

10 citations

Elizabeth Thomas, Retheesh S. Thankan, V. F. Rudchenko, Guangfei Huang, Vincent C.O. Njar +1 more

Targeted Degradation of Androgen Receptor by VNPP433-3β in Castration-Resistant Prostate Cancer Cells Implicates Interaction with E3 Ligase MDM2 Resulting in Ubiquitin-Proteasomal Degradation

Cancers(2023)10.3390/cancers15041198

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0DataRank · unranked

17 citations

Retheesh S. Thankan, Puranik Purushottamachar, David J. Weber, Vincent C.O. Njar, Elizabeth Thomas

VNLG-152R and its deuterated analogs potently inhibit/repress triple/quadruple negative breast cancer of diverse racial origins in vitro and in vivo by upregulating E3 Ligase Synoviolin 1 (SYVN1) and inducing proteasomal degradation of MNK1/2

Frontiers in Oncology(2023)10.3389/fonc.2023.1240996

N/A

0DataRank · unranked

4 citations

Elizabeth Thomas, Puranik Purushottamachar, David J. Weber, Vidya P. Ramamurthy, Weiliang Huang +3 more

Salinization Dramatically Enhance the Anti-Prostate Cancer Efficacies of AR/AR-V7 and Mnk1/2 Molecular Glue Degraders, Galeterone and VNPP433-3β Which Outperform Docetaxel and Enzalutamide in CRPC CWR22Rv1 Xenograft Mouse Model

Bioorganic Chemistry(2023)10.1016/j.bioorg.2023.106700

N/A

0DataRank · unranked

11 citations

Elizabeth Thomas, Puranik Purushottamachar, David J. Weber, Vincent C.O. Njar, Retheesh S. Thankan

Murine toxicology and pharmacokinetics of lead next generation galeterone analog, VNPP433-3β

Steroids(2023)10.1016/j.steroids.2023.109184

N/A

0DataRank · unranked

9 citations

Retheesh S. Thankan, Puranik Purushottamachar, Jianxia Guo, Robert A. Parise, Jan H. Beumer +2 more