Thomas E. Prisinzano

NeuroscienceBiochemistry, Genetics and Molecular BiologyMedicine

Pilot corpus only

This score is computed over theSindex pilot corpus and does not cover the full scientific literature. Scores are relative to papers we have ingested — papers, authors, and institutions outside the pilot are not represented. Methodology.

Top 100%percentile

0Author DataRank

Indexed papers

0in pilot corpus

datarank_citation_only_1hop_v6· scope data_onlyMethodology

Papers

Driven by 28 papers. Top paper: “Strategies for Developing κ Opioid Receptor Agonists for the Treatment of Pain with Fewer Side Effects”.

Strategies for Developing κ Opioid Receptor Agonists for the Treatment of Pain with Fewer Side Effects

Journal of Pharmacology and Experimental Therapeutics(2020)10.1124/jpet.120.000134

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55 citations

Diana Vivian Atigari, Sophia Kaska, Thomas E. Prisinzano, Bronwyn M. Kivell, Kelly F. Paton

G-Protein biased opioid agonists: 3-hydroxy- N -phenethyl-5-phenylmorphans with three-carbon chain substituents at C9

RSC Medicinal Chemistry(2020)10.1039/d0md00104j

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15 citations

Eric W. Bow, Fuying Li, Agnieszka Sulima, Sophia Kaska, Rachel Saylor Crowley +8 more

The Intriguing Effects of Substituents in the N-Phenethyl Moiety of Norhydromorphone: A Bifunctional Opioid from a Set of “Tail Wags Dog” Experiments

Molecules(2020)10.3390/molecules25112640

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12 citations

Thomas C. Irvin, Christine A. Herdman, Ramsey D. Hanna, Sergio A. Hassan, Yong Sok Lee +16 more

Synthetic Studies of Neoclerodane Diterpenes from Salvia divinorum: Design, Synthesis, and Evaluation of Analogues with Improved Potency and G-protein Activation Bias at the μ-Opioid Receptor

ACS Chemical Neuroscience(2020)10.1021/acschemneuro.0c00191

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31 citations

Andrew P. Riley, Amy F. Alder, R. J. Anderson, Dan Luo, Sophia Kaska +4 more

Evidence for the Involvement of Dopamine Transporters in Behavioral Stimulant Effects of Modafinil

UNC Libraries(2020)10.17615/kxkp-hr07

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7 citations

V. Setola, M. H. Baumann, Thomas E. Prisinzano, J. S. Partilla, B. L. Roth +3 more

Behavioral and Physiological Effects of a Novel Kappa-Opioid Receptor-Based DREADD in Rats

UNC Libraries(2020)10.17615/sjhp-f785

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0 citations

Jennifer M. Bossert, Bruce T. Hope, Brandon K. Harvey, Thomas E. Prisinzano, Yavin Shaham +6 more

Design, synthesis, and preliminary evaluation of a potential synthetic opioid rescue agent

Journal of Biomedical Science(2021)10.1186/s12929-021-00758-y

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20 citations

Dan Luo, Sophia Kaska, Kumar Kulldeep Niloy, Karen S. Jackson, R.J. Sarma +7 more

The Salvinorin Analogue, Ethoxymethyl Ether Salvinorin B, Promotes Remyelination in Preclinical Models of Multiple Sclerosis

Frontiers in Neurology(2021)10.3389/fneur.2021.782190

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18 citations

Katharina Robichon, Nikki Templeton, Lisa Denny, Afnan Al Abadey, Dan Luo +4 more

Profile of a short-acting κ-antagonist, LY2795050, on self-grooming behaviors, forced swim test and locomotor activity: sex comparison in mice

Journal of Psychopharmacology(2021)10.1177/0269881121996883

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9 citations

Caroline Baynard, Bryan D. McElroy, Thomas E. Prisinzano, Mary Jeanne Kreek, Eduardo R. Butelman

Rapid-Onset Anti-Stress Effects of a Kappa-Opioid Receptor Antagonist, LY2795050, Against Immobility in an Open Space Swim Paradigm in Male and Female Mice

Frontiers in Pharmacology(2021)10.3389/fphar.2021.775317

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2 citations

Thomas E. Prisinzano, Eduardo R. Butelman, Caroline Baynard

Discriminative-Stimulus Effects of Synthetic Cathinones in Squirrel Monkeys

The International Journal of Neuropsychopharmacology(2021)10.1093/ijnp/pyab017

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6 citations

Alexander M. Sherwood, Thomas E. Prisinzano, Jack Bergman, Stephen J. Kohut, Carol A. Paronis +1 more

Rational inhibitor design for Pseudomonas aeruginosa salicylate adenylation enzyme PchD

JBIC Journal of Biological Inorganic Chemistry(2022)10.1007/s00775-022-01941-8

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15 citations

Kathleen M. Meneely, Trey A. Ronnebaum, Annemarie S. Chilton, Andrew P. Riley, Thomas E. Prisinzano +2 more

A Journey through Diastereomeric Space: The Design, Synthesis, In Vitro and In Vivo Pharmacological Activity, and Molecular Modeling of Novel Potent Diastereomeric MOR Agonists and Antagonists

Molecules(2022)10.3390/molecules27196455

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11 citations

Agnieszka Sulima, Dan Luo, Thomas E. Prisinzano, Alexander Goldberg, Bing Xie +9 more

Synthesis and Pharmacological Evaluation of Enantiopure N-Substituted Ortho-c Oxide-Bridged 5-Phenylmorphans

Molecules(2022)10.3390/molecules27248808

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1 citations

Theresa Kopajtic, Jonathan L. Katz, Dan Luo, Thomas E. Prisinzano, Gregory H. Imler +4 more

Xylazine suppresses fentanyl consumption during self-administration and induces a unique sex-specific withdrawal syndrome that is not altered by naloxone in rats.

Experimental and Clinical Psychopharmacology(2023)10.1037/pha0000670

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42 citations

Safiyah Sadek, Percell Kendrick, Emma O. Bondy, Mei Hong, Sally Pauss +8 more

Discovery of a Potent Highly Biased MOR Partial Agonist among Diastereomeric C9-Hydroxyalkyl-5-phenylmorphans

Molecules(2023)10.3390/molecules28124795

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16 citations

Agnieszka Sulima, Eugene S. Gutman, Eric W. Bow, Dan Luo, Sophia Kaska +8 more

The Kappa Opioid Receptor Agonist 16-Bromo Salvinorin A Has Anti-Cocaine Effects without Significant Effects on Locomotion, Food Reward, Learning and Memory, or Anxiety and Depressive-like Behaviors

Molecules(2023)10.3390/molecules28124848

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10 citations

Amy Ewald, Susan Welsh, Lindsay Kornberger, Samuel E. Williamson, Bryan D. McElroy +4 more

A MOR Antagonist with High Potency and Antagonist Efficacy among Diastereomeric C9-Alkyl-Substituted N-Phenethyl-5-(3-hydroxy)phenylmorphans

Molecules(2023)10.3390/molecules28145411

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4 citations

Agnieszka Sulima, Dan Luo, Thomas E. Prisinzano, Arthur E. Jacobson, Kenner C. Rice +1 more

Potent MOR Agonists from 2′-Hydroxy-5,9-dimethyl-N-phenethyl Substituted-6,7-benzomorphans and from C8-Hydroxy, Methylene and Methyl Derivatives of N-Phenethylnormetazocine

Molecules(2023)10.3390/molecules28237709

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2 citations

George W. Ward, Agnieszka Sulima, Dan Luo, Thomas E. Prisinzano, Gregory H. Imler +4 more

Xylazine co-self-administration suppresses fentanyl consumption during self-administration and induces a unique sex-specific withdrawal syndrome that is not altered by naloxone in rats

bioRxiv (Cold Spring Harbor Laboratory)(2023)10.1101/2023.05.17.541158

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3 citations

Safiyah Sadek, Percell Kendrick, Emma O. Bondy, Mei Hong, Sally Pauss +8 more

Searching for Synthetic Opioid Rescue Agents: Identification of a Potent Opioid Agonist with Reduced Respiratory Depression

Journal of Medicinal Chemistry(2024)10.1021/acs.jmedchem.4c00333

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7 citations

Dan Luo, Kai Johnson, Emily D. Denehy, Judy C. Songrady, Jocelyn Martin +15 more

Targeting α1- and α2-adrenergic receptors as a countermeasure for fentanyl-induced locomotor and ventilatory depression

Environmental Toxicology and Pharmacology(2024)10.1016/j.etap.2024.104527

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7 citations

Emily D. Denehy, Jocelyn Martin, Cassie M. Chandler, Dan Luo, Chase E. Taylor +6 more

Functional Activity of Enantiomeric Oximes and Diastereomeric Amines and Cyano Substituents at C9 in 3-Hydroxy-N-phenethyl-5-phenylmorphans

Molecules(2024)10.3390/molecules29091926

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2 citations

Madhurima Das, Agnieszka Sulima, Dan Luo, Sophia Kaska, Thomas E. Prisinzano +4 more

Effects of Biased Analogues of the Kappa Opioid Receptor Agonist, U50,488, in Preclinical Models of Pain and Side Effects

Molecules(2025)10.3390/molecules30030604

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10 citations

Loan Y. Vu, Lindsay Kornberger, Dan Luo, Brittany Scouller, Sheein Hong +4 more

Preclinical Pharmacokinetic Evaluation of Mithramycin and Mithramycin SA Tryptophan-Conjugated Analog

Pharmaceutics(2025)10.3390/pharmaceutics17060765

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2 citations

Jamie Horn, Nazmul H. Bhuiyan, Khaled A. Shaaban, Suhas S. Bhosale, Thomas E. Prisinzano +4 more

Transformation of a Potent C9-Substituted Phenylmorphan into MOR Partial Agonists with Improvement of Metabolic Stability: An In Vitro, In Vivo, and In Silico Study

ACS Chemical Neuroscience(2025)10.1021/acschemneuro.5c00211

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1 citations

Dan Luo, Thomas E. Prisinzano, S. Stevens Negus, Nima Nassehi, Dana E. Selley +10 more

Searching for Synthetic Opioid Rescue Agents. 2: Identification of an Ultra-Potent Synthetic Opioid Rescue Agent

Journal of Medicinal Chemistry(2025)10.1021/acs.jmedchem.5c01108

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1 citations

Edem K. Onyameh, Dan Luo, Joshua W. Powell, Riya Trivedi, Eric J. Woloshin +12 more

N-(3-Hydroxyphenyl)-3,8-diazabicyclooctanes as opioid receptors probes. 1. Investigation of the phenolic hydroxyl group

European Journal of Medicinal Chemistry(2025)10.1016/j.ejmech.2025.117991

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0 citations

Dan Luo, Marissa C. Hessing, Emily Prantzalos, Warren J. Alilain, Jill Turner +2 more