John A. Katzenellenbogen

Biochemistry, Genetics and Molecular BiologyMedicineComputer ScienceChemistry

Pilot corpus only

This score is computed over theSindex pilot corpus and does not cover the full scientific literature. Scores are relative to papers we have ingested — papers, authors, and institutions outside the pilot are not represented. Methodology.

Top 100%percentile

0Author DataRank

Indexed papers

0in pilot corpus

datarank_citation_only_1hop_v6· scope data_onlyMethodology

Papers

Driven by 35 papers. Top paper: “The quest for improving the management of breast cancer by functional imaging: The discovery and development of 16α-[18F]fluoroestradiol (FES), a PET radiotracer for the estrogen receptor, a historical review”.

The quest for improving the management of breast cancer by functional imaging: The discovery and development of 16α-[18F]fluoroestradiol (FES), a PET radiotracer for the estrogen receptor, a historical review

Nuclear Medicine and Biology(2020)10.1016/j.nucmedbio.2020.02.007

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61 citations

John A. Katzenellenbogen

A mutant form of ERα associated with estrogen insensitivity affects the coupling between ligand binding and coactivator recruitment

Science Signaling(2020)10.1126/scisignal.aaw4653

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14 citations

Laurel A. Coons, René Houtman, Kathryn E. Carlson, Teresa A. Martin, Christopher G. Mayne +6 more

The tissue-specific effects of different 17β-estradiol doses reveal the key sensitizing role of AF1 domain in ERα activity

Molecular and Cellular Endocrinology(2020)10.1016/j.mce.2020.110741

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12 citations

Mélissa Buscato, Alexia Vinel, Frank Giton, Isabelle Raymond‐Letron, Sung Hoon Kim +9 more

Suppression of breast cancer metastasis and extension of survival by a new antiestrogen in a preclinical model driven by mutant estrogen receptors

Breast Cancer Research and Treatment(2020)10.1007/s10549-020-05629-y

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11 citations

Yvonne Ziegler, Sayyed Hamed Shahoei, Parama Dey, Sung Hoon Kim, Mayuri A. Yasuda +6 more

PET Imaging Agents (FES, FFNP, and FDHT) for Estrogen, Androgen, and Progesterone Receptors to Improve Management of Breast and Prostate Cancers by Functional Imaging

Cancers(2020)10.3390/cancers12082020

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30 citations

John A. Katzenellenbogen

Long-Term Follow-Up and Treatment of a Female With Complete Estrogen Insensitivity

The Journal of Clinical Endocrinology & Metabolism(2020)10.1210/clinem/dgaa106

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6 citations

Lynn P. Chorich, Hyung‐Goo Kim, Laurel A. Coons, John A. Katzenellenbogen, Janet E. Hall +3 more

VAV3 mediates resistance to breast cancer endocrine therapy

UNC Libraries(2020)10.17615/39pm-cr73

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0 citations

Olle Stål, Miguel Gil‐Gil, Laia Gómez‐Baldó, Xosé R. Bustelo, Xavier Barril +40 more

Radiosynthesis and Evaluation of Talazoparib and Its Derivatives as PARP-1-Targeting Agents

Biomedicines(2021)10.3390/biomedicines9050565

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27 citations

Huaping Chen, Cedric Mpoy, Sadia Afrin, Buck E. Rogers, Joel R. Garbow +3 more

Exploration of alcohol‐enhanced Cu‐mediated radiofluorination toward practical labeling

Journal of Labelled Compounds and Radiopharmaceuticals(2021)10.1002/jlcr.3955

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11 citations

Wenhua Chu, John A. Katzenellenbogen, Dong Zhou

Defining the Energetic Basis for a Conformational Switch Mediating Ligand-Independent Activation of Mutant Estrogen Receptors in Breast Cancer

Molecular Cancer Research(2021)10.1158/1541-7786.mcr-20-1017

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13 citations

Weiyi Toy, Kathryn E. Carlson, Trusha Bhatt, Sean W. Fanning, Geoffrey L. Greene +5 more

A simple method to generate [18F]triflyl fluoride for 18F radiosynthesis

Tetrahedron Letters(2021)10.1016/j.tetlet.2021.153273

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7 citations

John A. Katzenellenbogen, Dong Zhou

Determination of molar activity of [18F]fluoride by HPLC via sulfonyl derivatization

Applied Radiation and Isotopes(2021)10.1016/j.apradiso.2021.109865

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4 citations

Sally W. Schwarz, John A. Katzenellenbogen, Dong Zhou

Dual-mechanism estrogen receptor inhibitors

Proceedings of the National Academy of Sciences(2021)10.1073/pnas.2101657118

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0 citations

J.C. Nwachukwu, Charles K. Min, Jacqline W. Njeri, Sathish Srinivasan, Erumbi S. Rangarajan +16 more

CHRM1 is a Druggable Melanoma Target Whose Endogenous Activity is Determined by Inherited Genetic Variation in DOPA Production

bioRxiv (Cold Spring Harbor Laboratory)(2021)10.1101/2021.03.03.433757

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0 citations

Christopher A. Natale, In Young Lee, Swati Venkat, Sung Hoon Kim, John A. Katzenellenbogen +4 more

Estrogen Receptor Beta 1: A Potential Therapeutic Target for Female Triple Negative Breast Cancer

Endocrinology(2022)10.1210/endocr/bqac172

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17 citations

Alexander Wang, Yvonne Ziegler, Sandeep Kumar, Shunchao Yan, Sung Hoon Kim +3 more

Solid phase radiosynthesis of an olaparib derivative using 4-[18F] fluorobenzoic acid and in vivo evaluation in breast and prostate cancer xenograft models for PARP-1 expression

Nuclear Medicine and Biology(2022)10.1016/j.nucmedbio.2022.09.002

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5 citations

Huaping Chen, Buck E. Rogers, John A. Katzenellenbogen, Dong Zhou, Jinbin Xu

New 1,1-diarylethylene FOXM1 inhibitors potently reduce intracellular FOXM1 and suppress high-grade serous ovarian carcinoma cell viability

Research Square(2022)10.21203/rs.3.rs-1281554/v1

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2 citations

Catalina Muñoz-Trujillo, Sung Hoon Kim, John A. Katzenellenbogen, Benita S. Katzenellenbogen, Adam R. Karpf +1 more

Targeting the oncogenic transcription factor FOXM1 to improve outcomes in all subtypes of breast cancer

Breast Cancer Research(2023)10.1186/s13058-023-01675-8

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88 citations

Valeria Sanabria Guillen, John A. Katzenellenbogen, Benita S. Katzenellenbogen

ESR1 F404 Mutations and Acquired Resistance to Fulvestrant in ESR1 -Mutant Breast Cancer

Cancer Discovery(2023)10.1158/2159-8290.cd-22-1387

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38 citations

Alex Pearson, María Teresa Herrera-Abreu, Li-Xuan Sim, Rosalind Cutts, Heena Shah +12 more

Endothelial ERα promotes glucose tolerance by enhancing endothelial insulin transport to skeletal muscle

Nature Communications(2023)10.1038/s41467-023-40562-w

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24 citations

Ken L. Chambliss, Jun Peng, Jose Barrera, Keiji Tanigaki, Katherine Luby‐Phelps +14 more

[18F]Tosyl fluoride as a versatile [18F]fluoride source for the preparation of 18F-labeled radiopharmaceuticals

Scientific Reports(2023)10.1038/s41598-023-30200-2

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9 citations

Wenhua Chu, Jinbin Xu, Sally W. Schwarz, John A. Katzenellenbogen, Dong Zhou

Stringing along the estrogen receptor to engage with DNA

Proceedings of the National Academy of Sciences(2023)10.1073/pnas.2300608120

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4 citations

John A. Katzenellenbogen

NB compounds are potent and efficacious FOXM1 inhibitors in high-grade serous ovarian cancer cells

Journal of Ovarian Research(2024)10.1186/s13048-024-01421-4

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11 citations

Makenzie Vorderbruggen, Catalina Muñoz-Trujillo, Sung Hoon Kim, John A. Katzenellenbogen, Benita S. Katzenellenbogen +2 more

Iterative Catalyst-Controlled Diastereoselective Matteson Homologations Enable the Selective Synthesis of Benzestrol Isomers

Journal of the American Chemical Society(2024)10.1021/jacs.4c12857

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11 citations

Hayden A. Sharma, Chan K. Choi, Kathryn E. Carlson, Yingwei Hou, J.C. Nwachukwu +6 more

Asymmetric allostery in estrogen receptor-α homodimers drives responses to the ensemble of estrogens in the hormonal milieu

Proceedings of the National Academy of Sciences(2024)10.1073/pnas.2321344121

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7 citations

J.C. Nwachukwu, Yingwei Hou, Robin Russo, Alexandra Papa, Jian Min +9 more

Resistance to FOXM1 inhibitors in breast cancer is accompanied by impeding ferroptosis and apoptotic cell death

Breast Cancer Research and Treatment(2024)10.1007/s10549-024-07420-9

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6 citations

Yvonne Ziegler, Blake N. Plotner, Kristen M. Flatt, Sung Hoon Kim, John A. Katzenellenbogen +2 more

Asymmetric Allostery in Estrogen Receptor-α Homodimers Drives Responses to the Ensemble of Estrogens in the Hormonal Milieu

bioRxiv (Cold Spring Harbor Laboratory)(2024)10.1101/2024.04.10.588871

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0 citations

J.C. Nwachukwu, Yingwei Hou, Robin Russo, Alexandra Papa, Jian Min +9 more

Inhibition of FOXM1 synergizes with BCL2 inhibitor Venetoclax in killing non-t(11;14) multiple myeloma cells via repressing MYC pathway

bioRxiv (Cold Spring Harbor Laboratory)(2024)10.1101/2024.09.27.613548

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0 citations

Siegfried Janz, Yidan Wang, Benita S. Katzenellenbogen, John A. Katzenellenbogen, Sung Hoon Kim +2 more

Phthalates Impair Estrogenic Regulation of HIF2α and Extracellular Vesicle Secretion by Human Endometrial Stromal Cells

bioRxiv (Cold Spring Harbor Laboratory)(2024)10.1101/2024.12.12.628185

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0 citations

Arpita Bhurke, Kathryn E. Carlson, John A. Katzenellenbogen, Jie Yu, Jodi A. Flaws +3 more

Benzestrol Isomer Stereochemistry Determines the Distinct Estrogenic Activities and Conformations of the Eight Isomers When Bound to Estrogen Receptor α

ACS Pharmacology & Translational Science(2025)10.1021/acsptsci.5c00117

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2 citations

J.C. Nwachukwu, Kathryn E. Carlson, Sung Hoon Kim, Steven R. Angle, Eric N. Jacobsen +8 more

Targeting FOXM1 reshapes antitumor immunity to attenuate small cell lung cancer progression

Cancer Letters(2025)10.1016/j.canlet.2025.218160

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2 citations

Parvez Κhan, Mahek Fatima, Asad Rehman, Laiba Anwar, Zahraa Wajih Alsafwani +13 more

Phthalates Impair Estrogenic Regulation of HIF2α and Extracellular Vesicle Secretion by Human Endometrial Stromal Cells

Endocrinology(2025)10.1210/endocr/bqaf087

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3 citations

Arpita Bhurke, Kathryn E. Carlson, John A. Katzenellenbogen, Jie Yu, Jodi A. Flaws +3 more

Inhibition of FOXM1 Synergizes with BH3 Mimetics Venetoclax and Sonrotoclax in Killing Multiple Myeloma Cells through Repressing MYC Pathway

Advanced Science(2025)10.1002/advs.202508822

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3 citations

Yidan Wang, Kathryn Fox, Adam Bissonnette, Luke F. Moat, Terrie Kitchner +12 more

FOXM1 targeting alters AURKB activity and reshapes antitumor immunity to curb the progression of small cell lung cancer

Research Square(2025)10.21203/rs.3.rs-6960266/v1

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0 citations

Parvez Κhan, Mahek Fatima, Asad Rehman, Laiba Anwar, Zahraa Wajih Alsafwani +14 more

Chloroindazole based estrogen receptor β ligands with favorable pharmacokinetics promote functional remyelination and visual recovery

Scientific Reports(2025)10.1038/s41598-025-20254-9

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0 citations

Sung Hoon Kim, Flor de Fátima Rosas‐Cárdenas, Alyssa A. Anderson, B. Poole, D H Deshpande +15 more