Dilip K. Tosh

Also affiliated with National Institute of Diabetes and Digestive and Kidney Diseases

Biochemistry, Genetics and Molecular BiologyMedicineNeuroscience

Pilot corpus only

This score is computed over theSindex pilot corpus and does not cover the full scientific literature. Scores are relative to papers we have ingested — papers, authors, and institutions outside the pilot are not represented. Methodology.

Top 100%percentile

0Author DataRank

Indexed papers

0in pilot corpus

datarank_citation_only_1hop_v6· scope data_onlyMethodology

Papers

Driven by 28 papers. Top paper: “Structure of the human dopamine transporter and mechanisms of inhibition”.

Structure of the human dopamine transporter and mechanisms of inhibition

Nature(2024)10.1038/s41586-024-07739-9

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0.606DataRank · unranked

56 citations

Vikas Navratna, Dilip K. Tosh, Audrey Chinn, Md Fulbabu Sk, Emad Tajkhorshid +3 more

Design and in vivo activity of A3 adenosine receptor agonist prodrugs

Purinergic Signalling(2020)10.1007/s11302-020-09715-0

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0.449DataRank · unranked

19 citations

Shanu Jain, Zhoumou Chen, Dilip K. Tosh, Yanling Ma, Maren C. Podszun +4 more

Effects of Purinergic Receptor Deletion or Pharmacologic Modulation on Pulmonary Inflammation in Mice

ACS Pharmacology & Translational Science(2022)10.1021/acsptsci.2c00128

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0.373DataRank · unranked

11 citations

Tadeusz Karcz, Dilip K. Tosh, Kwan‐Young Jung, Zhiwei Wen, Ryan G. Campbell +5 more

A3 adenosine receptor agonists containing dopamine moieties for enhanced interspecies affinity

European Journal of Medicinal Chemistry(2021)10.1016/j.ejmech.2021.113983

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0.360DataRank · unranked

10 citations

Veronica Salmaso, Ryan G. Campbell, Harsha Rao, Amelia Bitant, Eline Pottie +7 more

Acute visceral pain relief mediated by A3AR agonists in rats: involvement of N-type voltage-gated calcium channels

Pain(2020)10.1097/j.pain.0000000000001905

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0DataRank · unranked

28 citations

Elisabetta Coppi, Laura Micheli, Carmen Parisio, Alessia Vona, Federica Cherchi +13 more

Nucleotide P2Y1 receptor agonists are in vitro and in vivo prodrugs of A1/A3 adenosine receptor agonists: implications for roles of P2Y1 and A1/A3 receptors in physiology and pathology

Purinergic Signalling(2020)10.1007/s11302-020-09732-z

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0DataRank · unranked

25 citations

Sonja Hinz, Christa E. Müller, Deborah Holstein, Jay M. Wendling, Roger J. Melton +9 more

Structure activity relationship of novel antiviral nucleosides against Enterovirus A71

Bioorganic & Medicinal Chemistry Letters(2020)10.1016/j.bmcl.2020.127599

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0DataRank · unranked

6 citations

Kiran S. Toti, Brett L. Hurst, Justin G. Julander, Kenneth A. Jacobson, Dilip K. Tosh

Pyrimidine Ribonucleotides with Enhanced Selectivity as P2Y 6 Receptor Agonists: Novel 4-Alkyloxyimino, (S)-Methanocarba, and 5′-Triphosphate γ-Ester Modifications †

UNC Libraries(2020)10.17615/9vwt-ya70

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0DataRank · unranked

0 citations

Barkın Berk, Kenneth A. Jacobson, Рамачандран Баласубраманиан, Dilip K. Tosh, Hiroshi Maruoka +6 more

Polyamidoamine (PAMAM) Dendrimer Conjugates of “Clickable” Agonists of the A 3 Adenosine Receptor and Coactivation of the P2Y 14 Receptor by a Tethered Nucleotide

UNC Libraries(2020)10.17615/wk9d-zk24

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0DataRank · unranked

0 citations

Zhan Gao, Matthew O. Barrett, Kenneth A. Jacobson, T. Kendall Harden, Ingrid Fricks +5 more

Adenosine A3 agonists reverse neuropathic pain via T cell–mediated production of IL-10

Journal of Clinical Investigation(2021)10.1172/jci139299

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0DataRank · unranked

69 citations

Silvia Squillace, Filomena Lauro, Luigino Antonio Giancotti, Elisabetta Coppi, Federica Cherchi +12 more

Optical control of adenosine A3 receptor function in psoriasis

Pharmacological Research(2021)10.1016/j.phrs.2021.105731

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0DataRank · unranked

25 citations

Ingrid Filgaira, Ernest G. Nolen, Gisela Cabré, Jordi Hernando, Dilip K. Tosh +4 more

Expanding the repertoire of methanocarba nucleosides from purinergic signaling to diverse targets

RSC Medicinal Chemistry(2021)10.1039/d1md00167a

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0DataRank · unranked

14 citations

Veronica Salmaso, R. Rama Suresh, Dilip K. Tosh, Kenneth A. Jacobson

Targeting the A3 adenosine receptor to prevent and reverse chemotherapy-induced neurotoxicities in mice

Acta Neuropathologica Communications(2022)10.1186/s40478-022-01315-w

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0DataRank · unranked

46 citations

Rajasekaran Mahalingam, Silvia Squillace, Kenneth A. Jacobson, Dilip K. Tosh, Shruti Dharmaraj +5 more

Interaction of A3 adenosine receptor ligands with the human multidrug transporter ABCG2

European Journal of Medicinal Chemistry(2022)10.1016/j.ejmech.2022.114103

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0DataRank · unranked

8 citations

Megumi Murakami, Dilip K. Tosh, Jinha Yu, Sabrina Lusvarghi, Ryan G. Campbell +4 more

First Potent Macrocyclic A3 Adenosine Receptor Agonists Reveal G-Protein and β-Arrestin2 Signaling Preferences

ACS Pharmacology & Translational Science(2023)10.1021/acsptsci.3c00126

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0DataRank · unranked

4 citations

Courtney Fisher, Veronica Salmaso, Tina C. Wan, Ryan G. Campbell, Eric Chen +4 more

2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A1 Adenosine Receptor Positive Allosteric Modulators

ACS Medicinal Chemistry Letters(2023)10.1021/acsmedchemlett.3c00315

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0DataRank · unranked

1 citations

R. Rama Suresh, Silvia Pasquini, Veronica Salmaso, E.J. Will, Dilip K. Tosh +7 more

Structure activity relationships of 5-HT2B and 5-HT2C serotonin receptor antagonists: N6, C2 and 5′-Modified (N)-methanocarba-adenosine derivatives

European Journal of Medicinal Chemistry(2023)10.1016/j.ejmech.2023.115691

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0DataRank · unranked

3 citations

Maggie M. Calkins, Marko Ivancich, Hailey A. Bock, Ryan G. Campbell, Sarah A. Lewicki +5 more

Photoswitchable Diazocine Derivative for Adenosine A3 Receptor Activation in Psoriasis

Journal of the American Chemical Society(2024)10.1021/jacs.4c13558

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0DataRank · unranked

23 citations

Mirko Scortichini, Dilip K. Tosh, Veronica Salmaso, Tongil Ko, Glòria Salort +7 more

Mitochondrial A3Adenosine Receptor as a Mechanism for the Protective Effects of A3AR Agonists on Chemotherapy-Induced Neuropathic Pain

Journal of Neuroscience(2024)10.1523/jneurosci.1268-24.2024

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0DataRank · unranked

11 citations

Kali Janes, Wen Xiao, Grant R. Kolar, Hans Luecke, Michael Anne Gratton +5 more

Potent and Selective Human 5-HT2B Serotonin Receptor Antagonists: 4′-Cyano-(N)-methanocarba-adenosines by Synthetic Serendipity

Journal of Medicinal Chemistry(2024)10.1021/acs.jmedchem.4c02174

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0DataRank · unranked

7 citations

Matteo Pavan, A. Clark, Josie Lammers, Serafina Villano, Silvia Marri +17 more

Selective modulation of epileptic tissue by an adenosine A3 receptor‐activating drug

British Journal of Pharmacology(2024)10.1111/bph.17319

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0DataRank · unranked

6 citations

Leonor Ribeiro‐Rodrigues, Gabriele Ruffolo, Veronica Alfano, Cátia Domingos, Nádia Rei +16 more

2-Substituted (N)-Methanocarba A3 Adenosine Receptor Agonists: In Silico, In Vitro, and In Vivo Characterization

ACS Pharmacology & Translational Science(2024)10.1021/acsptsci.4c00223

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0DataRank · unranked

8 citations

Matteo Pavan, Chunxia Cronin, Eline Pottie, Tina C. Wan, Eric Chen +8 more

Genetic and functional modulation by agonist MRS5698 and allosteric enhancer LUF6000 at the native A3 adenosine receptor in HL-60 cells

Purinergic Signalling(2024)10.1007/s11302-024-09992-z

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0DataRank · unranked

4 citations

Weiping Chen, Ray R. Gao, Jonathan Li, Dilip K. Tosh, John A. Hanover +2 more

Direct Comparison of (N)-Methanocarba and Ribose-Containing 2-Arylalkynyladenosine Derivatives as A3 Receptor Agonists

ACS Medicinal Chemistry Letters(2020)10.1021/acsmedchemlett.9b00637

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0DataRank · unranked

23 citations

Veronica Salmaso, Harsha Rao, Ryan G. Campbell, Amelia Bitant, Zhan‐Guo Gao +3 more

(N)-Methanocarba-adenosines as monoamine transporter allosteric inhibitors: Extended N6 groups for bitopic stabilization

European Journal of Medicinal Chemistry(2025)10.1016/j.ejmech.2025.118167

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0DataRank · unranked

0 citations

Matteo Pavan, Laura B. Kozell, Amy J. Eshleman, Jennifer L. Schmachtenberg, Katherine M. Wolfrum +4 more

Truncated (N)-Methanocarba Nucleosides as Partial Agonists at Mouse and Human A3 Adenosine Receptors: Affinity Enhancement by N6-(2-Phenylethyl) Substitution

Journal of Medicinal Chemistry(2020)10.1021/acs.jmedchem.0c00235

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0DataRank · unranked

20 citations

Veronica Salmaso, Harsha Rao, Amelia Bitant, Courtney Fisher, David I. Lieberman +7 more

Assessment of biased agonism at the A3 adenosine receptor using β-arrestin and miniGαi recruitment assays

Biochemical Pharmacology(2020)10.1016/j.bcp.2020.113934

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0DataRank · unranked

43 citations

Dilip K. Tosh, Zhan‐Guo Gao, Kenneth A. Jacobson, Christophe P. Stove, Eline Pottie

Chronic Morphine-Induced Changes in Signaling at the A3 Adenosine Receptor Contribute to Morphine-Induced Hyperalgesia, Tolerance, and Withdrawal

Journal of Pharmacology and Experimental Therapeutics(2020)10.1124/jpet.120.000004

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0DataRank · unranked

39 citations

Tally M. Largent‐Milnes, Zhoumou Chen, Vasiliki Staikopoulos, Emanuela Esposito, Rebecca Dalgarno +10 more